Bilastine 40 mg

Allergies are a common health concern affecting millions of people worldwide. Symptoms like sneezing, runny nose, nasal congestion, itching, and hives can interfere with daily life, productivity, and overall well-being. BISALATIN 40, containing Bilastine 40 mg, is a second-generation, non-sedating antihistamine designed to provide effective and lasting relief from allergic symptoms.

With its once-daily dosing, non-sedating profile, and high efficacy, BISALATIN 40 has become a preferred choice for adults and adolescents dealing with seasonal allergic rhinitis, perennial rhinitis, and chronic urticaria.

Composition

Each BISALATIN 40 tablet contains:

• Bilastine 40 mg: The active ingredient responsible for reducing allergic symptoms by blocking H1 histamine receptors.

Inactive ingredients (excipients) may include: microcrystalline cellulose, lactose monohydrate, magnesium stearate, colloidal silicon dioxide, and other binders and coatings that ensure the tablet’s stability, absorption, and ease of use.

How BISALATIN 40 Works

Bilastine 40 mg works by blocking H1 histamine receptors in the body. Histamine is a chemical released by the immune system during an allergic reaction, causing itching, sneezing, watery eyes, and hives. By preventing histamine from binding to these receptors, BISALATIN 40 alleviates allergy symptoms effectively.

• Peripheral Action: Bilastine acts mainly on peripheral tissues such as the skin, nose, and respiratory tract.

• Non-Sedating: Minimal penetration into the central nervous system ensures that patients remain alert and active.

• Rapid Onset: Relief typically starts within 1–2 hours, lasting up to 24 hours with a single dose.

Uses of BISALATIN 40

BISALATIN 40 is prescribed for:

• Seasonal allergic rhinitis (hay fever): Reduces sneezing, nasal congestion, runny nose, and watery eyes.

• Perennial allergic rhinitis: Controls year-round allergy symptoms caused by dust, pollen, or pet dander.

• Chronic urticaria: Helps reduce itching, redness, and hives, providing significant symptom relief.

It is suitable for adults and adolescents aged 12 years and above, offering convenient, once-daily dosing.

Benefits of BISALATIN 40

1. Non-Sedating Formula: Unlike first-generation antihistamines, BISALATIN 40 does not cause drowsiness, allowing patients to carry on daily activities safely.

2. Once-Daily Convenience: Simplifies treatment and improves adherence.

3. Fast-Acting Relief: Symptoms are relieved within 1–2 hours.

4. Long-Lasting Effect: Provides 24-hour relief, reducing the need for multiple doses.

5. Effective for Multiple Allergy Types: Works for both rhinitis and urticaria, making it a versatile solution.

6. Well-Tolerated: Minimal side effects compared to older antihistamines.

Dosage

• Adults and Adolescents (12 years and above): Take 1 tablet of BISALATIN 40 mg once daily.

• Timing: Ideally on an empty stomach (1 hour before or 2 hours after meals) for optimal absorption.

• Children under 12: Use only under medical supervision.

Important: Follow the prescribed dosage. Do not exceed recommended amounts without consulting a healthcare provider.

Side Effects

BISALATIN 40 is generally well-tolerated. Some patients may experience mild side effects, including:

• Headache

• Dizziness

• Mild gastrointestinal discomfort

• Rare allergic reactions such as rash or swelling

Most users experience no significant side effects, and the non-sedating nature ensures minimal interference with daily activities.

Precautions

• Pregnancy & Breastfeeding: Consult a healthcare provider before use.

• Medical Conditions: Patients with kidney or liver issues should seek medical advice.

• Medication Interactions: Inform your doctor if you are taking other medications, especially other antihistamines or antifungal drugs.

• Allergies: Avoid BISALATIN 40 if allergic to bilastine or any other component of the tablet.

• Storage: Store in a cool, dry place, away from direct sunlight and moisture. Keep out of reach of children.

How Does Bilastine 40 mg Work in the Body?

Bilastine 40 mg is a second-generation antihistamine widely used to treat allergic conditions such as seasonal allergic rhinitis, perennial rhinitis, and chronic urticaria. Unlike first-generation antihistamines, Bilastine is non-sedating and provides effective allergy relief without causing drowsiness, making it suitable for daily use in adults and children.

Mechanism of Action

Bilastine works by blocking H1 histamine receptors in the body. Histamine is a chemical released by the immune system in response to allergens, causing symptoms like sneezing, itching, runny nose, watery eyes, and hives.

• H1 Receptor Antagonism: Bilastine selectively binds to peripheral H1 receptors found in the skin, nose, and respiratory tract. By blocking these receptors, it prevents histamine from causing allergic reactions.

• Peripheral Action: Unlike older antihistamines, Bilastine has minimal penetration into the central nervous system (CNS). This reduces sedation and allows the patient to remain alert during daily activities.

Onset and Duration of Action

• Rapid Relief: Bilastine 40 mg typically starts working within 1–2 hours after oral intake.

• Long-Lasting Effect: A single dose provides 24-hour relief from allergy symptoms, making it convenient for once-daily dosing.

Clinical Effects in the Body

1. Respiratory Tract:

   • Reduces sneezing, nasal congestion, and runny nose caused by allergic rhinitis.

   • Eases nasal itching and watery discharge during seasonal or perennial allergies.

2. Skin:

   • Alleviates itching, redness, and hives in chronic urticaria.

   • Prevents the formation of new hives by inhibiting histamine-induced inflammation.

3. Eye Symptoms:

   • Reduces itching, redness, and tearing associated with ocular allergies.

Advantages of Bilastine 40 mg

• Non-Sedating: Patients can take it during the day without drowsiness.

• Once-Daily Dosing: Convenient and ensures consistent symptom control.

• Safe for Adults and Children: Recommended in age-appropriate doses with minimal side effects.

• Minimal Drug Interactions: Safe to use with other common medications like decongestants or painkillers.

Who Can Benefit from Bilastine 40 mg?

• Individuals suffering from seasonal allergies caused by pollen, dust, or animal dander.

• Patients with perennial allergic rhinitis triggered by indoor allergens.

• People experiencing chronic urticaria (hives) with itching, redness, and swelling.

• Individuals who need effective allergy relief without sedation.

What is the Composition of Bilastine Tablets?

Bilastine tablets are a widely used second-generation antihistamine designed to relieve allergy symptoms such as sneezing, runny nose, itching, and hives. The effectiveness of Bilastine comes from its carefully formulated active and inactive ingredients, which ensure targeted action, minimal side effects, and better absorption. Understanding its composition helps in appreciating how this medicine provides fast and reliable relief from allergic reactions.

Active Ingredient

• Bilastine 40 mg: The primary active component in the tablet is Bilastine, which belongs to the class of H1 receptor antagonists.

  • Function: Bilastine works by blocking H1 histamine receptors, preventing histamine from triggering allergic symptoms such as sneezing, itching, hives, and watery eyes.

  • Dose: Each tablet typically contains 40 mg of Bilastine, which is suitable for once-daily dosing in adults and adolescents.

Inactive Ingredients (Excipients)

The inactive ingredients in Bilastine tablets help in maintaining the tablet’s stability, absorption, and shelf life. Common excipients include:

• Microcrystalline cellulose: Provides structural integrity to the tablet.

• Lactose monohydrate: Used as a filler to ensure consistent tablet weight.

• Magnesium stearate: Acts as a lubricant to prevent sticking during manufacturing.

• Colloidal silicon dioxide: Enhances tablet flow and prevents caking.

• Other binders and coatings: Ensure easy swallowing, stability, and controlled dissolution.

Note: The exact list of excipients may vary slightly depending on the manufacturer or brand, but the active ingredient (Bilastine 40 mg) remains consistent.

Mechanism of Action Related to Composition

• The active ingredient Bilastine directly targets peripheral H1 receptors, reducing histamine-mediated symptoms without significant central nervous system penetration, which makes it non-sedating.

• The inactive ingredients support tablet integrity, absorption, and patient compliance, ensuring that Bilastine is delivered effectively in the body.

Benefits of the Composition

• Fast-Acting Relief: The active ingredient works quickly to relieve sneezing, runny nose, and itching.

• Non-Sedating: Bilastine’s selective H1 receptor action ensures daytime alertness.

• Once-Daily Dose: 40 mg per tablet allows for convenient, simple dosing.

• Safe and Stable: Inactive ingredients help maintain tablet stability, shelf life, and efficacy.

• Minimal Side Effects: Carefully selected excipients reduce the risk of digestive discomfort.

Who Can Use Bilastine Tablets?

• Adults and adolescents (12 years and above): For relief of seasonal and perennial allergic rhinitis.

• Patients with chronic urticaria: Helps reduce itching, redness, and hives.

• Individuals needing non-sedating antihistamines: Safe for daily activities without causing drowsiness.

Common FAQs About Bilastine 40 mg Tablets

Bilastine 40 mg is a second-generation, non-sedating antihistamine commonly prescribed for allergic rhinitis, chronic urticaria, and other allergy-related conditions. Patients often have questions regarding its uses, dosage, safety, and effectiveness. This FAQ guide addresses the most frequently asked questions, helping users make informed decisions.

1. What is Bilastine 40 mg?

Bilastine 40 mg is a prescription antihistamine used to relieve allergy symptoms such as sneezing, runny nose, itching, and hives. It works by blocking H1 histamine receptors in the body, preventing the effects of histamine without causing sedation.

2. What is Bilastine used for?

Bilastine tablets are primarily used for:

• Seasonal allergic rhinitis (hay fever)

• Perennial allergic rhinitis (year-round allergies)

• Chronic urticaria (persistent hives)

It helps reduce itching, redness, swelling, sneezing, and watery eyes.

3. How does Bilastine work in the body?

Bilastine works by selectively blocking peripheral H1 histamine receptors, which prevents histamine from causing allergy symptoms. Unlike older antihistamines, it does not significantly enter the central nervous system, making it non-drowsy.

4. How should Bilastine 40 mg be taken?

• Adults and adolescents (12 years and above): Take one tablet (40 mg) once daily.

• Timing: Ideally, take it on an empty stomach (1 hour before or 2 hours after food) for optimal absorption.

• Do not exceed the prescribed dose without consulting a doctor.

5. When does Bilastine start working?

Bilastine usually starts working within 1–2 hours of oral intake, providing 24-hour relief from allergy symptoms. Continuous daily use ensures consistent symptom control.

6. Is Bilastine 40 mg safe during pregnancy or breastfeeding?

• Pregnancy: Only use under the guidance of a healthcare provider.

• Breastfeeding: Limited data is available, so consultation with a doctor is advised before use.

7. What are the side effects of Bilastine 40 mg?

Bilastine is generally well-tolerated. Common side effects may include:

• Mild headache

• Dizziness

• Stomach discomfort
  Rarely, some may experience allergic reactions such as rash or swelling. Most people experience no significant side effects, especially compared to first-generation antihistamines.

8. Can Bilastine cause drowsiness?

Bilastine is a non-sedating antihistamine. Most patients do not experience drowsiness, making it safe to use during the day without affecting work or driving.

9. Can Bilastine be taken with other medications?

Bilastine has minimal drug interactions. However, consult your doctor if you are taking:

• Other antihistamines

• Heart medications

• Antifungal drugs or strong inhibitors of P-glycoprotein

Always inform your doctor about all medications and supplements before starting Bilastine.

10. Who should avoid taking Bilastine 40 mg?

• Individuals with allergy to Bilastine or any component of the tablet

• Patients with severe kidney impairment

• People advised by their doctor to avoid antihistamines due to specific medical conditions

11. Can Bilastine be used for children?

• Bilastine is generally prescribed for children aged 12 and above.

• Pediatric dosing and safety should always follow doctor recommendations.

12. How long can Bilastine 40 mg be used?

• Short-term use: For seasonal allergy relief, usually for a few days to weeks.

• Long-term use: Can be used for chronic urticaria under medical supervision.

• Important: Do not self-medicate for prolonged periods without consulting a healthcare professional.

13. How should Bilastine tablets be stored?

• Store in a cool, dry place away from direct sunlight.

• Keep out of reach of children.

• Avoid exposure to moisture to maintain tablet effectiveness.

14. Can Bilastine 40 mg be purchased over-the-counter in India?

Bilastine is prescription-only in India, so a doctor’s consultation is usually required before purchase to ensure safe and appropriate use.

15. Why choose Bilastine 40 mg over other antihistamines?

• Non-sedating: Allows patients to stay alert.

• Once-daily dosing: Convenient for daily use.

• Fast onset: Symptom relief starts in 1–2 hours.

• Well-tolerated: Minimal side effects compared to older antihistamines.